反应条件
sodium tetrahydroborate; triphenylphosphine; trifluoroacetic acid; Wang resin; diethylazodicarboxylate 1.) THF, 24 h, RT; 2.) CH2Cl2, H2O, 90 min, RT; 3.) CH2Cl2, RT, 30 min; Yield givenMultistep reaction;
参考文献
Tetrahedron Letters, , vol. 40, # 24 p. 4535 - 4538