反应条件
1: K2CO3 / N,N-dimethyl-acetamide / 2 h / 170 °C
2: MgSO4 / toluene / 100 °C
3: cesium pivalate / Pd(OAc)2; 1,1-bis(diphenylphosphino)methane / dimethylformamide / 24 h / 100 °C
4: aq. HCl / acetone
View Scheme
参考文献
Zhao, Jian; Yue, Dawei; Campo, Marino A.; Larock, Richard C.
Journal of the American Chemical Society, 2007 , vol. 129, # 16 p. 5288 - 5295