(1-重氮-2-氧代-丙醇)-膦酸二甲酯合成路线

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参考文献

Wijtmans, Maikel; De Graaf, Chris; De Kloe, Gerdien; Istyastono, Enade P.; Smit, Judith; Lim, Herman; Boonnak, Ratchanok; Nijmeijer, Saskia; Smits, Rogier A.; Jongejan, Aldo; Zuiderveld, Obbe; De Esch, Iwan J. P.; Leurs, Rob
Journal of Medicinal Chemistry, 2011 , vol. 54, # 6 p. 1693 - 1703

941-55-9对甲苯磺酰叠氮+

4202-14-6丙酮基膦酸二甲酯

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90965-06-3(1-重氮-2-氧代-丙醇)-膦酸二甲酯

参考文献

SCHERING CORPORATION
Patent: WO2007/97937 A1, 2007 ;
Location in patent: Page/Page column 190 ;
WO 2007/097937 A1

4202-14-6丙酮基膦酸二甲酯+

2158-14-74-乙酰氨基苯磺酰叠氮

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90965-06-3(1-重氮-2-氧代-丙醇)-膦酸二甲酯

参考文献

Helvetica Chimica Acta, , vol. 88, # 11 p. 2918 - 2937

90965-06-3(1-重氮-2-氧代-丙醇)-膦酸二甲酯+

20949-84-22-甲基-1,3-噻唑-4-甲醛

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107263-89-84-乙炔-2-甲基噻唑

参考文献

Paterson, Ian; Menche, Dirk; Hakansson, Anders E.; Longstaff, Adrian; Wong, David; Barasoain, Isabel; Buey, Ruben M.; Diaz, J. Fernando
Bioorganic and Medicinal Chemistry Letters, 2005 , vol. 15, # 9 p. 2243 - 2247

90965-06-3(1-重氮-2-氧代-丙醇)-膦酸二甲酯+

120-14-93,4-二甲氧基苯甲醛

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4302-52-73,4-二甲氧基苯乙炔

参考文献

Koufaki, Maria; Theodorou, Elissavet; Galaris, Dimitrios; Nousis, Lambros; Katsanou, Efrosini S.; Alexis, Michael N.
Journal of Medicinal Chemistry, 2006 , vol. 49, # 1 p. 300 - 306

90965-06-3(1-重氮-2-氧代-丙醇)-膦酸二甲酯+

4707-71-59-甲醛菲

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32870-98-79-乙炔基菲

参考文献

Synlett, , # 19 p. 3037 - 3041

3029-19-41-芘甲醛+

90965-06-3(1-重氮-2-氧代-丙醇)-膦酸二甲酯

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34993-56-11-乙炔基芘

参考文献

Maisonneuve, Stephane; Xie, Juan
Synlett, 2009 , # 18 p. 2977 - 2981