反应条件
1: 77 percent / K2CO3 / acetone / 24 h / Heating
2: 1.) TiCl4, 2.) 1 N aq. HCl / 1.) a) CH2Cl2, 0 deg C, 1 h, b) RT, 4 h
View Scheme
参考文献
Langlois, Michel; Bremont, Beatrice; Shen, Shuren; Poncet, Annie; Andrieux, Jean; et al.
Journal of Medicinal Chemistry, 1995 , vol. 38, # 12 p. 2050 - 2060