1.1: sodium hydride / N,N-dimethyl-formamide; mineral oil / 6 h / 0 - 20 °C / Inert atmosphere 1.2: 20 °C / Inert atmosphere 2.1: caesium carbonate / water; methanol / 1 h / 20 °C View Scheme
参考文献
BRITISH COLUMBIA CANCER AGENCY BRANCH; THE UNIVERSITY OF BRITISH COLUMBIA; SADAR, Marianne D.; MAWJI, Nasrin R.; BANUELOS, Carmen Adriana; ANDERSEN, Raymond J.; GARCIA FERNANDEZ, Javier
Patent: WO2011/82487 A1, 2011 ;
WO 2011/082487 A1