反应条件
1: 1.) 15 percent BuLi / 1.) hexane, THF, 0 deg C, 2.) 30 min 2: 68 percent / CH3I, CaCO3 / methanol; H2O / 20 h / Heating View Scheme
参考文献
Hofmeister; Annen; Laurent; Petzoldt; Wiechert
Arzneimittel-Forschung/Drug Research, 1986 , vol. 36, # 5 p. 781 - 783