反应条件
1: With tetrachloromethane; 4-(N,N-dimethlyamino)pyridine; N-ethyl-N,N-diisopropylamine in acetonitrile
T=23°C; 1 h;
2: With trifluoroacetic acid in dichloromethane
0.5 h;
参考文献
Deprez, Pierre; Mandine, Eliane; Gofflo, Dominique; Meunier, Stephane; Lesuisse, Dominique
Bioorganic and Medicinal Chemistry Letters, 2002 , vol. 12, # 9 p. 1295 - 1298