1: With toluene-4-sulfonic acid in water; acetonitrile
T=0 - 10°C; 0.166667 h;
2: With sodium azide; sodium nitrite in water
T=10 - 15°C; 0.166667 h;
3: With sodium azide
参考文献
Qi, Jianjun; Tung, Ching-Hsuan
Bioorganic and Medicinal Chemistry Letters, 2011 , vol. 21, # 1 p. 320 - 323