1: furan-2-ylmethylamine With sodium hydride in tetrahydrofuran; mineral oil 6 h; Inert atmosphere; 2: 3-chloropropanoyl chloride in tetrahydrofuran; mineral oil T=20°C; Inert atmosphere;
参考文献
Bodill, Taryn; Conibear, Anne C.; Mutorwa, Marius K.M.; Goble, Jessica L.; Blatch, Gregory L.; Lobb, Kevin A.; Klein, Rosalyn; Kaye, Perry T.
Bioorganic and Medicinal Chemistry, 2013 , vol. 21, # 14 p. 4332 - 4341