反应条件
1: With potassium carbonate in N,N-dimethyl-formamide T=0 - 20°C; Inert atmosphere; 2: in N,N-dimethyl-formamide T=60°C; 5.5 h;
参考文献
Niculescu-Duvaz, Dan; Niculescu-Duvaz, Ion; Suijkerbuijk, Bart M.J.M.; Menard, Delphine; Zambon, Alfonso; Davies, Lawrence; Pons, Jean-Francois; Whittaker, Steven; Marais, Richard; Springer, Caroline J.
Bioorganic and Medicinal Chemistry, 2013 , vol. 21, # 5 p. 1284 - 1304