反应条件
1: 1.) NaH / 1.) DMF, 25 deg C, 1 h, 2.) DMF, RT, 15 h 2: 89 percent / triethylamine / toluene / 1.) reflux, 8 h, 2.) RT, 15 h View Scheme
参考文献
Malleron, Jean-Luc; Comte, Marie-Therese; Gueremy, Claude; Peyronel, Jean Francois; Truchon, Alain; et al.
Journal of Medicinal Chemistry, 1991 , vol. 34, # 8 p. 2477 - 2483