1: With 4-(N,N-dimethlyamino)pyridine in dichloromethane T=0 - 5°C; 2: With dicyclohexyl-carbodiimide in dichloromethane T=0 - 20°C; Product distribution / selectivity;
参考文献
RAMOT AT TEL AVIV UNIVERSITY LTD.; BAR-ILAN UNIVERSITY; BIOLINERX LTD.
Patent: WO2006/131923 A2, 2006 ;
Location in patent: Page/Page column 47 ;