反应条件
1: triethylamine / CH2Cl2 / Ambient temperature
2: diborane / tetrahydrofuran / a) RT, 1 h, b) reflux, 90 min
3: 95 percent / KOH / aq. ethanol / 5 h / Heating
View Scheme
参考文献
Albright; DeVries; Largis; Miner; Reich; Schaffer; Shepherd; Upeslacis
Journal of Medicinal Chemistry, 1983 , vol. 26, # 10 p. 1378 - 1393