2-(4-甲基苯基)-1H-吲哚合成路线 （共 57 条）
反应条件
oxygen; acetic acid; palladium diacetate
T=20°C; P=760.051 Torr; 10 h;
参考文献
Yang, Shang-Dong; Sun, Chang-Liang; Fang, Zhao; Li, Bi-Jie; Li, Yi-Zhou; Shi, Zhang-Jie
Angewandte Chemie - International Edition, 2008 , vol. 47, # 8 p. 1473 - 1476
反应条件
5 Au/Fe2O3; hydrogen in toluene
T=60 - 120°C; P=750.075 - 15001.5 Torr; 2 h; Autoclave; chemoselective reaction;
参考文献
Yamane, Yoshihiro; Liu, Xiaohao; Hamasaki, Akiyuki; Ishida, Tamao; Haruta, Masatake; Yokoyama, Takushi; Tokunaga, Makoto
Organic Letters, 2009 , vol. 11, # 22 p. 5162 - 5165
反应条件
[Fe(II)(C5H5)(C5H4PPh2)]; gold monoiodide; potassium carbonate in toluene
T=130°C; Sonogashira reaction; 24 h;
参考文献
Li, Pinhua; Wang, Lei; Wang, Min; You, Feng
European Journal of Organic Chemistry, 2008 , # 35 p. 5946 - 5951
反应条件
Au/Carbon G-60 catalyst (0.5 percent wt, 5.3 mg) in toluene
T=90°C; 24 h; Inert atmosphereSchlenk technique; Reagent/catalystTemperature;
参考文献
Perea-Buceta, Jesus E.; Wirtanen, Tom; Laukkanen, Otto-Ville; Maekelae, Mikko K.; Nieger, Martin; Melchionna, Michele; Huittinen, Nina; Lopez-Sanchez, Jose A.; Helaja, Juho
Angewandte Chemie - International Edition, 2013 , vol. 52, # 45 p. 11835 - 11839
Angew. Chem., 2013 , vol. 125, # 45 p. 12051 - 12055,5
反应条件
rhodium(II) heptafluorobutyrate in toluene
T=60°C; 16 h; Molecular sieve;
参考文献
Shen, Meihua; Leslie, Brooke E.; Driver, Tom G.
Angewandte Chemie - International Edition, 2008 , vol. 47, # 27 p. 5056 - 5059
反应条件
cobalt/rhodium in tetrahydrofuran
T=90°C; P=15201 Torr; 5 h;
参考文献
Park, Ji Hoon; Kim, Eunha; Chung, Young Keun
Organic Letters, 2008 , vol. 10, # 21 p. 4718 - 4721
反应条件
palladium diacetate; magnesium oxide; triphenylphosphine in 1,4-dioxane; N,N-dimethyl-formamide
T=150°C; 18 h;
参考文献
Sezen, Bengue; Sames, Dalibor
Journal of the American Chemical Society, 2003 , vol. 125, # 18 p. 5274 - 5275
反应条件
dicyclohexyl(2′,6′-dimethoxybiphenyl-2-yl)phosphine; potassium phosphate; palladium diacetate in toluene
T=90°C; 5 h;
参考文献
Fang, Yuan-Qing; Lautens, Mark
Journal of Organic Chemistry, 2008 , vol. 73, # 2 p. 538 - 549
反应条件
n-butyllithium in tetrahydrofuran; hexane
T=20°C;
参考文献
Primofiore, Giampaolo; Da Settimo, Federico; Taliani, Sabrina; Simorini, Francesca; Patrizi, Maria Paola; Novellino, Ettore; Greco, Giovanni; Abignente, Enrico; Costa, Barbara; Chelli, Beatrice; Martini, Claudia
Journal of Medicinal Chemistry, 2004 , vol. 47, # 7 p. 1852 - 1855
反应条件
sodium t-butanolate; 2-(dicyclohexylphosphino)-2',4',6'-tri-i-propyl-1,1’-biphenyl; tris-(dibenzylideneacetone)dipalladium(0) in toluene
T=110°C; Heck reaction; 20 h;
参考文献
Barluenga, Jose; Fernandez, M. Alejandro; Aznar, Fernando; Valdes, Carlos
Chemistry - A European Journal, 2005 , vol. 11, # 8 p. 2276 - 2283
