反应条件
1: 1,1'-carbonyldiimidazole; magnesium chloride / tetrahydrofuran / 50 °C
2: 1,8-diazabicyclo[5.4.0]undec-7-ene / ethanol / 80 °C
View Scheme
参考文献
Fukunaga, Kenji; Uehara, Fumiaki; Aritomo, Keiichi; Shoda, Aya; Hiki, Shinsuke; Okuyama, Masahiro; Usui, Yoshihiro; Watanabe, Kazutoshi; Yamakoshi, Koichi; Kohara, Toshiyuki; Hanano, Tokushi; Tanaka, Hiroshi; Tsuchiya, Susumu; Sunada, Shinji; Saito, Ken-Ichi; Eguchi, Jun-Ichi; Yuki, Satoshi; Asano, Shoichi; Tanaka, Shinji; Mori, Akiko; Yamagami, Keiji; Baba, Hiroshi; Horikawa, Takashi; Fujimura, Masatake
Bioorganic and Medicinal Chemistry Letters, 2013 , vol. 23, # 24 p. 6933 - 6937