3-乙酰胺基苯硼酸频哪醇酯合成路线 (共 5 条)
反应条件
potassium acetate; (1,1'-bis(diphenylphosphino)ferrocene)palladium(II) dichloride in 1,4-dioxane T=85°C; Inert atmosphere;
参考文献
WO2011/130628 A1, ;
Page/Page column 169 ;
WO 2011/130628 A1
反应条件
NiCl2(PMe3)2; TMSOCH2CF3; cesium fluoride in 1,4-dioxane T=100°C; 12 h; Inert atmosphere;
参考文献
Organic Letters, , vol. 13, # 21 p. 5766 - 5769
参考文献
US2008/269523 A1, ;
Page/Page column 6 ;
反应条件
in dichloromethane T=20°C; 10 h;
参考文献
Heterocycles, , vol. 80, # 2 p. 1359 - 1376
反应条件
1: triethylamine / dichloromethane / 2 h / 0 °C 2: potassium acetate / (1,1'-bis(diphenylphosphino)ferrocene)palladium(II) dichloride / 1,4-dioxane / 85 °C / Inert atmosphere View Scheme
参考文献
WO2011/130628 A1, ;
WO 2011/130628 A1