1: 2-bromoethyl phosphorodichloridate; (+/-)-3-octadecanamido-2-ethoxy-1-propanol Alkylation; 2: trimethylamine With water in chloroform; N,N-dimethyl-formamide; isopropyl alcohol Amination;
参考文献
Liu, Dong-Zhou; Morris-Natschke, Susan L.; Kucera, Louis S.; Ishaq, Khalid S.; Thakker, Dhiren R.
Journal of Pharmaceutical Sciences, 1999 , vol. 88, # 11 p. 1169 - 1174