5-溴-3-氟吡啶合成路线

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Jaeschke, Georg; Kolczewski, Sabine; Porter, Richard Hugh Philip; Vieira, Eric
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625-92-33,5-二溴吡啶

407-20-55-溴-3-氟吡啶

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Yamada, Shigeyuki; Knochel, Paul
Synthesis, 2010 , # 14 art. no. T09010SS, p. 2490 - 2494

2546-52-33-氟-4-溴吡啶

372-47-43-氟吡啶+

407-20-55-溴-3-氟吡啶

参考文献

Mallet, M.; Queguiner, G.
Tetrahedron, 1986 , vol. 42, # 8 p. 2253 - 2262

407-20-55-溴-3-氟吡啶

452972-09-7

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VERTEX PHARMACEUTICALS INCORPORATED; MACIKENAS, Dainius
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407-20-55-溴-3-氟吡啶

872041-86-6

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Page/Page column 36-37 ;

557-21-1氰化锌+

407-20-55-溴-3-氟吡啶

696-42-4

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MERCK SHARP and DOHME CORP.; BENNETT, D. Jonathan; CAI, Jaiqiang; CARSWELL, Emma; COOKE, Andrew; HOYT, Scott, B.; LONDON, Clare; MACLEAN, John; RATCLIFFE, Paul; TAYLOR, Jerry Andrew; XIONG, Yusheng; SAMANTA, Swapan Kumar; KULKARNI, Bheemashankar, A.
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407-20-55-溴-3-氟吡啶+

74-88-4甲基碘

1211517-76-8

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Hoffmann-La Roche Inc.; Alam, Muzaffar; DuBois, Daisy Joe; Hawley, Ronald Charles; Kennedy-Smith, Joshua; Minatti, Ana Elena; Palmer, Wylie Solang; Silva, Tania; Thakkar, Kshitij Chhabilbhai; Wilhelm, Robert Stephen
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407-20-55-溴-3-氟吡啶+

75-03-6碘乙烷

1374655-69-2

参考文献

MERCK SHARP and DOHME CORP.; BENNETT, D. Jonathan; CAI, Jaiqiang; CARSWELL, Emma; COOKE, Andrew; HOYT, Scott, B.; LONDON, Clare; MACLEAN, John; PARK, Min, K.; RATCLIFFE, Paul; XIONG, Yusheng; SAMANTA, Swapan Kumar; KULKARNI, Bheemashankar, A.
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Location in patent: Page/Page column 37 ;

407-20-55-溴-3-氟吡啶+

541-41-3氯甲酸乙酯

1214335-25-7

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CHLORION PHARMA, INC.; UNIVERSITE LAVAL; ATTARDO, Giorgio; TRIPATHY, Sasmita
Patent: WO2010/132999 A1, 2010 ;
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407-20-55-溴-3-氟吡啶+

75-31-0异丙胺

1201643-57-3

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NOVARTIS AG; FURET, Pascal; IMBACH, Patricia; MAH, Robert; STAUFFER, Frederic
Patent: WO2010/139747 A1, 2010 ;
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WO 2010/139747 A1