1: With triphenylphosphine; diethylazodicarboxylate in tetrahydrofuran
T=20°C; Mitsunobu reaction;
2: With beta-hydroxyethylmercaptan; 1,8-diazabicyclo[5.4.0]undec-7-ene in acetonitrile
T=20°C;
参考文献
Congreve, Miles S.; Kay, Corinne; Scicinski, Jan J.; Ley, Steven V.; Williams, Geoffrey; Murray, Peter J.; McKeown, Stephen C.; Watson, Stephen P.
Tetrahedron Letters, 2003 , vol. 44, # 21 p. 4153 - 4156