反应条件
1: 1.) n-BuLi / 1.) hexane, THF, -110 deg C, 1.25 h, 2.) hexane, THF, -110 deg C, 0.1 h, RT, 16 h 2: 1.) SOCl2 / 1.) CH2Cl2, RT, 1 h, 2.) CH2Cl2, reflux, 0.25 h View Scheme
参考文献
Street; Baker; Book; Reeve; Saunders; Willson; Marwood; Patel; Freedman
Journal of Medicinal Chemistry, 1992 , vol. 35, # 2 p. 295 - 305