Terent'Ev, Alexander O.; Krylov, Igor B.; Timofeev, Vladimir P.; Starikova, Zoya A.; Merkulova, Valentina M.; Ilovaisky, Alexey I.; Nikishin, Gennady I.
Advanced Synthesis and Catalysis, 2013 , vol. 355, # 11-12 p. 2375 - 2390
1: With lithium hexamethyldisilazane in tetrahydrofuran T=-78°C; 0.75 h; Inert atmosphere; 2: With trifluoromethylsulfonic anhydride in tetrahydrofuran T=-78 - 20°C; Inert atmosphere; 3: With ammonium chloride in tetrahydrofuran; water T=20°C;
参考文献
Maity, Pradip; Lepore, Salvatore D.
Journal of Organic Chemistry, 2009 , vol. 74, # 1 p. 158 - 162
Timonen, Juri M.; Nieminen, Riina M.; Sareila, Outi; Goulas, Antonis; Moilanen, Lauri J.; Haukka, Matti; Vainiotalo, Pirjo; Moilanen, Eeva; Aulaskari, Paula H.
European Journal of Medicinal Chemistry, 2011 , vol. 46, # 9 p. 3845 - 3850