N-乙氧羰基-4-哌啶酮合成路线 （共 74 条）
反应条件
triethylamine in dichloromethane T=0 - 20°C; 2 h;
参考文献
SUVEN LIFE SCIENCES LIMITED; Nirogi, Ramakrishna; Mohammed, Abdul Rasheed; Yarlagadda, Suresh; Ravella, Srinivasa Rao; Shinde, Anil Karbhari; Kamphampati, Ramasastri; Roayapalley, Praveen Kumar; Jayarajan, Pradeep; Bhyrapuneni, Gopinadh; Patnala, Sriramachandra Murthy; Ravula, Jyothsna; Jasti, Venkateswarlu
Patent: US2014/187581 A1, 2014 ;
Location in patent: Paragraph 0195-0198 ;
反应条件
in benzene T=0 - 20°C;
参考文献
US2005/234046 A1, ;
Page/Page column 59 ;
US 20050234046 A1
反应条件
methanol; potassium carbonate in dichloromethane T=20°C;
参考文献
Bioorganic and Medicinal Chemistry Letters, , vol. 18, # 20 p. 5439 - 5442
反应条件
in benzene 5 h; Heating;
参考文献
Praliev, K. D.; Belikova, N. A.; Isin, Zh. I.; Sokolov, D. V.
Pharmaceutical Chemistry Journal, 1987 , vol. 21, # 1 p. 60 - 61
Khimiko-Farmatsevticheskii Zhurnal, 1987 , vol. 21, # 1 p. 70 - 71
反应条件
1: Et3N / CH2Cl2 2: 3N HCl View Scheme
参考文献
Tetrahedron Letters, , vol. 34, # 24 p. 3863 - 3866
参考文献
Tetrahedron Letters, , vol. 34, # 24 p. 3863 - 3866
参考文献
Tetrahedron Letters, , vol. 29, # 27 p. 3303 - 3306
反应条件
in ethanol Fischer Indole Synthesis; 3 h; Reflux;
参考文献
NATIONAL UNIVERSITY OF SINGAPORE; RAMANUJULU, Pondy Murugappan; YANG, Tianming; CASEY, Mei-Wang; CASEY, Patrick J; GO, Mei Lin
Patent: WO2013/180656 A1, 2013 ;
Location in patent: Paragraph 000135; 000136 ;
反应条件
in ethanol 1.75 h; Heating;
参考文献
Harbert, Charles A.; Plattner, Jacob J.; Welch, Willard M.; Weissman, Albert; Koe, B. Kenneth
Journal of Medicinal Chemistry, 1980 , vol. 23, # 6 p. 635 - 643
反应条件
acetic acid 3 h; Reflux;
参考文献
Bonjoch, Josep; Diaba, Faiza; Pages, Lluis; Perez, Daniel; Soca, Lidia; Miralpeix, Montserrat; Vilella, Dolors; Anton, Paquita; Puig, Carles
Bioorganic and Medicinal Chemistry Letters, 2009 , vol. 19, # 15 p. 4299 - 4302
