N-Boc-乙醇胺合成路线

参考文献

BIOGEN IDEC MA INC.; ERLANSON, Daniel, A.; MARCOTTE, Doug; KUMARAVEL, Gnanasambandam; FAN, Junfa; WANG, Deping; CUERVO, Julio, H.; SILVIAN, Laura; POWELL, Noel; BUI, Minna; HOPKINS, Brian, T.; TAVERAS, Art; GUAN, Bing; CONLON, Patrick; ZHONG, Min; JENKINS, Tracy, J.; SCOTT, Daniel; SUNESIS PHARMACEUTICALS, INC.; LUGOVSKOY, Alexey, A.
Patent: WO2011/29046 A1, 2011 ;
WO 2011/029046 A1

541-59-3马来酰亚胺+

26690-80-2N-Boc-乙醇胺

134272-63-2叔丁基 (2-(2,5-二氧代-2,5-二氢-1H-吡咯-1-基)乙基)氨基甲酸酯

参考文献

Antczak; Bauvois; Monneret; Florent
Bioorganic and Medicinal Chemistry Letters, 2001 , vol. 11, # 21 p. 2843 - 2848

26690-80-2N-Boc-乙醇胺+

79-11-8氯乙酸

142929-49-5Boc-5-氨基-3-氧杂戊酸

参考文献

MYREXIS, INC.; BAJJI, Ashok, C.; TANGALLAPALLY, Rajendra, P.; KIM, In, Chul; KIM, Se, Ho; PARKER, Daniel, P.; TROVATO, Richard; PAPAC, Damon, I.; YAGER, Kraig; BAICHWAL, Vijay, R.
Patent: WO2012/148550 A1, 2012 ;
Location in patent: Page/Page column 50; 51 ;

26690-80-2N-Boc-乙醇胺

142929-49-5Boc-5-氨基-3-氧杂戊酸

参考文献

Adamczyk, Maciej; Fishpaugh, Jeffrey R.; Thiruvazhi, Mohan
Organic Preparations and Procedures International, 2002 , vol. 34, # 3 p. 326 - 331

26690-80-2N-Boc-乙醇胺

141-43-5乙醇胺

参考文献

SMITHKLINE BEECHAM CORPORATION
Patent: WO2006/113837 A2, 2006 ;
Location in patent: Page/Page column 101-102 ;
WO 2006/113837 A2

24424-99-5二碳酸二叔丁酯+

26690-80-2N-Boc-乙醇胺+

1972-28-7偶氮二甲酸二乙酯

13036-02-75-羟基间苯二甲酸二甲酯

参考文献

Microcide Pharmaceuticals, Inc.; DAIICHI PHARMACEUTICAL CO., LTD.
Patent: EP1227084 A1, 2002 ;

26690-80-2N-Boc-乙醇胺+

98-59-9对甲苯磺酰氯

158690-56-32-([叔丁氧羰基]氨基)乙基 4-甲基苯磺酸酯

参考文献

McGouran, Joanna F.; Kramer, Holger B.; MacKeen, Mukram M.; Di Gleria, Katalin; Altun, Mikael; Kessler, Benedikt M.
Organic and Biomolecular Chemistry, 2012 , vol. 10, # 17 p. 3379 - 3383

26690-80-2N-Boc-乙醇胺

168892-66-84-(2-叔丁氧羰氨基乙氧基)-苯甲酸

参考文献

Duggan; Duong; Fisher; Hamill; Hoffman; Huff; Ihle; Leu; Nagy; Perkins; Rodan; Wesolowski; Whitman; Zartman; Hartman
Journal of Medicinal Chemistry, 2000 , vol. 43, # 20 p. 3736 - 3745

26690-80-2N-Boc-乙醇胺

113525-94-3

参考文献

Liu, Gang; Tai, Wan-Yi; Li, Yu-Lin; Nan, Fa-Jun
Tetrahedron Letters, 2006 , vol. 47, # 19 p. 3295 - 3298

26690-80-2N-Boc-乙醇胺

114326-10-2S-[2-({[(2-甲基-2-丙基)氧基]羰基}氨基)乙基]硫代乙酸酯

参考文献

Vedejs, E.; Stults, J. S.
Journal of Organic Chemistry, 1988 , vol. 53, # 10 p. 2226 - 2232