反应条件
1: 2-mercaptoethanamine hydrochloride With tetra-(n-butyl)ammonium iodide; caesium carbonate in N,N-dimethyl-formamide T=20°C; 12 h; 2: 2-bromo-ethylamine-hydrobromide in N,N-dimethyl-formamide T=0 - 20°C; 1 h;
参考文献
Salvatore, Ralph Nicholas; Smith, Robert A.; Nischwitz, Adam K.; Gavin, Terrence
Tetrahedron Letters, 2005 , vol. 46, # 51 p. 8931 - 8935