1: 4-chloro-1H-indole With tetra(n-butyl)ammonium hydrogensulfate; sodium hydroxide in dichloromethane; water 0.25 h; 2: p-toluenesulfonyl chloride in dichloromethane; water T=20°C; 3 h;
1: 4-chloro-1H-indole With sodium hydride in N,N-dimethyl-formamide
T=20°C; 1 h;
2: benzyl bromide in N,N-dimethyl-formamide
T=20°C; 20 h;
参考文献
Evans, David A.; Scheidt, Karl A.; Fandrick, Keith R.; Lam, Hon Wai; Wu, Jimmy
Journal of the American Chemical Society, 2003 , vol. 125, # 36 p. 10780 - 10781
