4'-溴-2'-甲基乙酰苯胺合成路线 (共 43 条)
反应条件
benzyltrimethylammonium chlorobromate in methanol; dichloromethane 10 h; Ambient temperature;
参考文献
Kajigaeshi, Shoji; Kakinami, Takaaki; Yamasaki, Hiromichi; Fujisaki, Shizuo; Okamoto, Tsuyoshi
Bulletin of the Chemical Society of Japan, 1988 , vol. 61, # 7 p. 2681 - 2683
反应条件
triethylamine in dichloromethane from 0 deg C to RT;
参考文献
Borror, Alan L.; Chinoporos, Efthimios; Filosa, Michael P.; Herchen, Stephen R.; Petersen, Cheryl Pizzo; Stern, Carol A.
Journal of Organic Chemistry, 1988 , vol. 53, # 9 p. 2047 - 2052
反应条件
triethylamine in dichloromethane T=0°C;
参考文献
Mikami, Masafumi; Shinkai, Seiji
Journal of the Chemical Society, Chemical Communications, 1995 , # 2 p. 153 - 154
反应条件
N-bromosuccinmide in tetrachloromethane 2.5 h; HeatingIrradiation;
参考文献
Collins, David J.; Drygala, Peter F.; Swan, John M.
Australian Journal of Chemistry, 1983 , vol. 36, # 10 p. 2095 - 2110
参考文献
Journal of the American Chemical Society, , vol. 35, p. 972
参考文献
Pfizer Inc.
Patent: US4762838 A1, 1988 ;
参考文献
Pfizer Inc.
Patent: US4762838 A1, 1988 ;
反应条件
in dichloromethane T=0 - 20°C;
参考文献
European Journal of Organic Chemistry, , vol. 2014, # 3 p. 564 - 574
参考文献
US6337351 B1, ;
Example 15 ;
反应条件
1: AcOH; NaOH 2: Br2 View Scheme
参考文献
Bioorganic and Medicinal Chemistry Letters, , vol. 17, # 7 p. 1860 - 1864