1: With lithium aluminium tetrahydride in diethyl ether T=20°C; 3.5 h; Heating / reflux; 2: With sodium hydroxide; water in diethyl ether T=20°C; 1.5 h; 3: With hydrogenchloride in diethyl ether
参考文献
AMGEN INC.
Patent: WO2009/73203 A1, 2009 ;
Location in patent: Page/Page column 67 ;
WO 2009/073203 A1