in diethyl ether 1) 0 deg C, 1 h 2) 4 deg C , overnight;
参考文献
Tadros, William M.; Awadallah, Raafat; Grigis, Nabih S.
Indian Journal of Chemistry, Section B: Organic Chemistry Including Medicinal Chemistry, 1980 , vol. 19, # 9 p. 815 - 816
Lin, Edward Yin-Shiang; Guckian, Kevin M.; Silvian, Laura; Chin, Donovan; Ann Boriack-Sjodin; van Vlijmen, Herman; Friedman, Jessica E.; Scott, Daniel M.
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Journal of Medicinal Chemistry, 1989 , vol. 32, # 6 p. 1147 - 1156
(i) aq. NaNO2, dioxane, (ii) nBu3N, Ph2CH2; Multistep reaction;
参考文献
New, James S.; Christopher, William L.; Yevich, Joseph P.; Butler, Rhett; Schlemmer, R. Francis; et al.
Journal of Medicinal Chemistry, 1989 , vol. 32, # 6 p. 1147 - 1156