N-乙酰基-3-吲哚啉酮合成路线 （共 51 条）
反应条件
(2S)-3-phenylpropane-1,2-diamine; trifluoroacetic acid in chloroform
T=30°C; Michael addition; 72 h; optical yield given as percent ee;
参考文献
Sun, Wangsheng; Hong, Liang; Wang, Rui
Chemistry - A European Journal, 2011 , vol. 17, # 22 p. 6030 - 6033
反应条件
1: 90 percent / p-TsOH / toluene / 5 h / Heating
2: 21 percent / ethane-1,2-diol / 10 h / Heating
View Scheme
参考文献
Tugusheva; Ryabova; Solov'eva; Anisimova; Granik
Chemistry of Heterocyclic Compounds, 2001 , vol. 37, # 7 p. 885 - 893
反应条件
in acetic acid
5 h; Heating;
参考文献
Tugusheva; Ryabova; Solov'eva; Anisimova; Granik
Chemistry of Heterocyclic Compounds, 2001 , vol. 37, # 7 p. 885 - 893
反应条件
molybdenum peroxide hexamethylphosphorylamide in dichloromethane
96 h; Ambient temperature;
参考文献
Chien, Chung-Sheng; Takanami, Toshikatsu; Kawasaki, Tomomi; Sakamoto, Masanori
Chemical & Pharmaceutical Bulletin, 1985 , vol. 33, # 5 p. 1843 - 1848
反应条件
piperidine
3.5 h; Heating;
参考文献
Velzheva, V. S.; Nevskii, K. V.; Suvorov, N. N.
Chemistry of Heterocyclic Compounds (New York, NY, United States), 1985 , vol. 21, # 2 p. 191 - 196
Khimiya Geterotsiklicheskikh Soedinenii, 1985 , vol. 21, # 2 p. 230 - 235
反应条件
piperidine in benzene
3.5 h;
参考文献
Velezheva, V. S.; Marshakov, V. Yu.; Mel'man, A. I.; Kurkovskaya, L. N.; Suvorov, N. N.
Journal of Organic Chemistry USSR (English Translation), 1988 , p. 1379 - 1387
Zhurnal Organicheskoi Khimii, 1988 , vol. 24, # 7 p. 1531 - 1540
反应条件
piperidine in acetic acid
24 h; Heating;
参考文献
Bergman, Jan; Tilstam, Ulf
Tetrahedron, 1985 , vol. 41, # 14 p. 2883 - 2884
反应条件
in toluene
4 h; Heating;
参考文献
Kawasaki; Nonaka; Uemura; Sakamoto
Synthesis, 1991 , # 9 p. 701 - 702
反应条件
1: 74 percent / benzene / 0.33 h / 50 °C
2: 84 percent / acetic acid / 1 h / Heating
View Scheme
参考文献
Merour, Jean-Yves; Savelon, Laurence
Heterocycles, 1991 , vol. 32, # 5 p. 849 - 853
反应条件
acetic acid
1 h; Heating; Mechanism;
参考文献
Merour, Jean-Yves; Savelon, Laurence
Heterocycles, 1991 , vol. 32, # 5 p. 849 - 853
