sodium hydrogencarbonate in tetrahydrofuran T=20 - 25°C; 48 h;
参考文献
Piper, James R.; DeGraw, Joseph I.; Colwell, William T.; Johnson, Cheryl A.; Smith, R. Lane; Waud, William R.; Sirotnak, Francis M.
Journal of Medicinal Chemistry, 1997 , vol. 40, # 3 p. 377 - 384