1: 61 percent / K2CO3 / H2O; tetrahydrofuran / 2 h / 20 °C 2: 97 percent / TEA; HOBt; EDCl / dimethylformamide / 5 h / 20 °C 3: 94 percent / TEA / methanol / 24 h / 60 °C View Scheme
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