1,2,3,4-四氢苯并[b]氮杂卓-5-酮合成路线

24310-36-91-(甲苯-4-磺酰基)-1,2,3,4-四氢苯并[b]氮杂卓-5-酮

参考文献

FERRING B.V.
Patent: WO2006/21213 A2, 2006 ;
Location in patent: Page/Page column 34 ;
WO 2006/021213 A2

参考文献

Tsunoda, Takashi; Yamazaki, Atsuki; Iwamoto, Hidenori; Sakamoto, Shuichi
Organic Process Research and Development, 2003 , vol. 7, # 6 p. 883 - 887

4641-57-01-苯基-2-吡咯烷酮

635-90-51-苯基吡咯+

1127-74-81,2,3,4-四氢苯并[b]氮杂卓-5-酮

参考文献

Heterocycles, , vol. 36, # 4 p. 743 - 749

1127-74-81,2,3,4-四氢苯并[b]氮杂卓-5-酮

1701-57-12,3,4,5-四氢-1H-苯并[b]氮杂卓

参考文献

HYDRA BIOSCIENCES, INC.
Patent: WO2006/122156 A2, 2006 ;
Location in patent: Page/Page column 125 ;
WO 2006/122156 A2

1127-74-81,2,3,4-四氢苯并[b]氮杂卓-5-酮

137976-09-11-（4-氨基苯甲酰基）-2,3,4,5-四氢苯并[b]氮杂卓-5-酮

参考文献

Tsunoda, Takashi; Yamazaki, Atsuki; Iwamoto, Hidenori; Sakamoto, Shuichi
Organic Process Research and Development, 2003 , vol. 7, # 6 p. 883 - 887

1127-74-81,2,3,4-四氢苯并[b]氮杂卓-5-酮+

98-59-9对甲苯磺酰氯

24310-36-91-(甲苯-4-磺酰基)-1,2,3,4-四氢苯并[b]氮杂卓-5-酮

参考文献

ELI LILLY AND COMPANY
Patent: WO2005/37796 A1, 2005 ;
Location in patent: Page/Page column 160 ;

1127-74-81,2,3,4-四氢苯并[b]氮杂卓-5-酮+

108-24-7乙酸酐

1206-74-2

参考文献

STERIX LIMITED
Patent: WO2007/3934 A2, 2007 ;
Location in patent: Page/Page column 237-238 ;
WO 2007/003934 A2

1127-74-81,2,3,4-四氢苯并[b]氮杂卓-5-酮

137976-61-51-[4-(2-甲基苯甲酰胺基)苯甲酰基]-5-氧代-2,3,4,5-四氢-1H-1-苯并氮杂卓

参考文献

Ogawa, Hidenori; Yamashita, Hiroshi; Kondo, Kazumi; Yamamura, Yoshitaka; Miyamoto, Hisashi; Kan, Keizo; Kitano, Kazuyoshi; Tanaka, Michinori; Nakaya, Kenji; Nakamura, Shigeki; Mori, Toyoki; Tominaga, Michiaki; Yabuuchi, Youichi
Journal of Medicinal Chemistry, 1996 , vol. 39, # 18 p. 3547 - 3555

1127-74-81,2,3,4-四氢苯并[b]氮杂卓-5-酮+

108-23-6氯甲酸异丙酯

851044-97-8

参考文献

ELI LILLY AND COMPANY
Patent: WO2005/37796 A1, 2005 ;
Location in patent: Page/Page column 39 ;

1127-74-81,2,3,4-四氢苯并[b]氮杂卓-5-酮+

4635-59-04-氯丁酰氯

855783-84-5

参考文献

ABBOTT GMBH and CO. KG
Patent: WO2005/56546 A1, 2005 ;
Location in patent: Page/Page column 63 ;
WO 2005/056546 A1