反应条件
1: polyphosphoric acid / benzene / Heating 2: 1.) t-BuLi / 1.) Et2O, -78 deg C, 2.) Et2O View Scheme
参考文献
Tasker, Andrew S.; Sorensen, Bryan K.; Jae, Hwan-Soo; Winn, Martin; Von Geldern, Thomas W.; Dixon, Douglas B.; Chiou, William J.; Dayton, Brian D.; Calzadila, Samuel; Hernandez, Lisa; Marsh, Kennan C.; WuWong, J. Ruth; Opgenorth, Terry J.
Journal of Medicinal Chemistry, 1997 , vol. 40, # 3 p. 322 - 330