反应条件
1: (R)-glycidyl p-toluenesulfonate; benzene-1,2-diol With potassium carbonate in N,N-dimethyl-formamide T=60°C; 22 h; 2: p-toluenesulfonyl chloride in N,N-dimethyl-formamide T=0 - 20°C; 20 h; 3: potassium phtalimide Further stages;
参考文献
McComsey, David F.; Smith-Swintosky, Virginia L.; Parker, Michael H.; Brenneman, Douglas E.; Malatynska, Ewa; White, H. Steve; Klein, Brian D.; Wilcox, Karen S.; Milewski, Michael E.; Herb, Mark; Finley, Michael F. A.; Liu, Yi; Lubin, Mary Lou; Qin, Ning; Reitz, Allen B.; Maryanoff, Bruce E.
Journal of Medicinal Chemistry, 2013 , vol. 56, # 22 p. 9019 - 9030
