1: NaN3 / dimethylformamide / Ambient temperature 2: 1.) hydrogen, 2.) HCl / Pd-C / ethanol / 3 h / 45 °C View Scheme
参考文献
Venuti, Michael C.; Alvarez, Robert; Bruno, John J.; Strosberg, Arthur M.; Gu, Leo; et al.
Journal of Medicinal Chemistry, 1988 , vol. 31, # 11 p. 2145 - 2152