反应条件
1: 1.) LiNH2 / 1.) THF, -78 deg C, 30 min, 2.) THF, RT, 16 h 2: 92 percent / NaI / acetone / 12 h / Heating 3: 69 percent / dimethylsulfoxide / 1 h / Ambient temperature 4: 71 percent / NaBH4, H2, Ni(OAc)2, ethylenediamine / aq. ethanol / 2.5 h View Scheme
参考文献
Journal of Labelled Compounds and Radiopharmaceuticals, , vol. 36, # 6 p. 599 - 609
