反应条件
1: bis(2-oxo-3-oxazolidinyl)phosphinic chloride, Et3N / 1,2-dichloro-ethane / 18 h / Ambient temperature 2: potassium hexamethyldisilazide / tetrahydrofuran; toluene / 1 h / Ambient temperature View Scheme
参考文献
Rowley, Michael; Kulagowski, Janusz J.; Watt, Alan P.; Rathbone, Denise; Stevenson, Graeme I.; Carling, Robert W.; Baker, Raymond; Marshall, George R.; Kemp, John A.; Foster, Alan C.; Grimwood, Sarah; Hargreaves, Richard; Hurley, Catherine; Saywell, Kay L.; Tricklebank, Mark D.; Leeson, Paul D.
Journal of Medicinal Chemistry, 1997 , vol. 40, # 25 p. 4053 - 4068