反应条件
1: diethyl cyanophosphate, Et3N / dimethylformamide / 4 h 2: POCl3, P2O5 / 2 h / Heating View Scheme
参考文献
Gray, Nancy M.; Cheng, Brian K.; Mick, Stephen J.; Lair, Cecelia M.; Contreras, Patricia C.
Journal of Medicinal Chemistry, 1989 , vol. 32, # 6 p. 1242 - 1248