反应条件
1: 43 percent / ammonium acetate / acetic acid / 15 h / 20 °C
2: 44 percent / NaBH4 / ethanol / 1.) 20 deg C, 1 h, 2.) 50 deg C, 20 min
3: 32 percent / sulfur / 1 h / 200 °C
View Scheme
参考文献
Mobio, I. G.; Soldatenkov, A. T.; Fedorov, V. O.; Ageev, E. A.; Sergeeva, N. D.; et al.
Pharmaceutical Chemistry Journal, 1989 , vol. 23, # 4 p. 308 - 314
Khimiko-Farmatsevticheskii Zhurnal, 1989 , vol. 23, # 4 p. 421 - 427