反应条件
aluminium trichloride; sodium amide
1.) -20 deg C, 1 h, 2.) NH3 (liq.), -70 deg C, 1 h; Yield given. Multistep reaction;
参考文献
Peters, Richard H.; Crowe, David F.; Tanabe, Masato; Avery, Mitchell A.; Chong, Wesley K. M.
Journal of Medicinal Chemistry, 1987 , vol. 30, # 4 p. 646 - 652