噻唑并[4,5-b]吡啶-2(3h)-硫酮合成路线 (共 3 条)
反应条件
1: in N,N-dimethyl-formamide T=130°C; 2: With hydrogenchloride in N,N-dimethyl-formamide T=20°C; 1 h;
参考文献
WO2007/146066 A2, ;
Page/Page column 92 ;
参考文献
Bioorganic and Medicinal Chemistry Letters, , vol. 19, # 21 p. 6176 - 6180
反应条件
potassium carbonate in N,N-dimethyl-formamide
T=0°C;
参考文献
Bethge, Lucas; Jarikote, Dilip Venkatrao; Seitz, Oliver
Bioorganic and Medicinal Chemistry, 2008 , vol. 16, # 1 p. 114 - 125