N-Boc-3-哌啶酮合成路线

85275-45-21-Boc-3-羟基哌啶→98977-36-7N-Boc-3-哌啶酮

参考文献

COATS, STEVEN J.; BIAN, HAIYAN; CONNOLLY, PETER J.; BIGNAN, GILLES; CAI, CHAOZHONG; DAX, SCOTT L.; DECORTE, BART L.; LIN, SHU-CHEN; LIU, LI; MACIELAG, MARK J.; PITIS, PHILIP M.; ZHANG, YUE-MEI; ZHU, BIN; HE, WEI
Patent: US2011/105520 A1, 2011 ;
Location in patent: Page/Page column 36 ;

40114-49-61-苄基-3-哌啶酮+34619-03-9→98977-36-7N-Boc-3-哌啶酮

参考文献

US2003/229094 A1, ;

Page 123 ;
US 20030229094 A1

79-37-8草酰氯+85275-45-21-Boc-3-羟基哌啶→98977-36-7N-Boc-3-哌啶酮

参考文献

Kubo, Keiji; Miyawaki, Toshio; Kawamura, Masaki
Patent: US2003/187023 A1, 2003 ;

1179348-67-4→98977-36-7N-Boc-3-哌啶酮

参考文献

Mangion, Ian K.; Nwamba, Ikenna K.; Shevlin, Michael; Huffman, Mark A.
Organic Letters, 2009 , vol. 11, # 16 p. 3566 - 3569

24424-99-5二碳酸二叔丁酯+50717-82-33-哌啶酮→98977-36-7N-Boc-3-哌啶酮

参考文献

Journal of Medicinal Chemistry, , vol. 29, # 2 p. 224 - 229

114615-82-6过钌酸四丙胺盐(TPAP)+7529-22-8N-甲基吗啉氮氧化物→98977-36-7N-Boc-3-哌啶酮

参考文献

US2004/19058 A1, ;
US 20040019058 A1

6859-99-03-羟基哌啶→98977-36-7N-Boc-3-哌啶酮

参考文献

US5902882 A1, ;

85275-45-21-Boc-3-羟基哌啶+87413-09-0戴斯-马丁氧化剂→

参考文献

Bridger, Gary; Kaller, Al; Harwig, Curtis; Skerlj, Renato; Bogucki, David; Wilson, Trevor R.; Crawford, Jason; McEachern, Ernest J.; Atsma, Bem; Nan, Siqiao; Zhou, Yuanxi; Schols, Dominique; Smith, Christopher D.; Di Fluri, Maria R.
Patent: US2004/19058 A1, 2004 ;
US 20040019058 A1

24424-99-5二碳酸二叔丁酯→98977-36-7N-Boc-3-哌啶酮

参考文献

Emmett, George C.; Cain, Gary A.; Estrella, Melissa J.; Holler, Edd R.; Piecara, James S.; Blum, Andrew M.; Mical, Alfred J.; Teleha, Christopher A.; Wacker, Dean A.
Synthesis, 2005 , # 1 art. no. M04304SS, p. 92 - 96

6859-99-03-羟基哌啶→98977-36-7N-Boc-3-哌啶酮

参考文献

Bioorganic and Medicinal Chemistry, , vol. 15, # 1 p. 350 - 364