2,4-二氯-8-氟喹唑啉合成路线 (共 3 条)
反应条件
1: With acetic acid in water T=35°C; 3 h; 2: With N,N-dimethyl-aniline; trichlorophosphate T=130°C; 5 h;
参考文献
US2008/255156 A1, ;
Page/Page column 10 ;
反应条件
1: aq. AcOH / 2 h 2: POCl3, N,N-diethylaniline / 5 h / Heating View Scheme
参考文献
Journal of Medicinal Chemistry, , vol. 38, # 14 p. 2763 - 2773
反应条件
N,N-diethylaniline; trichlorophosphate 5 h; Heating;
参考文献
Journal of Medicinal Chemistry, , vol. 38, # 14 p. 2763 - 2773