1-[(4-苄基氧基苯基)-(二甲基氨基甲酰)甲基]环己醇合成路线 (共 1 条)
反应条件
1: With borane-THF in tetrahydrofuran T=0°C; 3.33 h; Heating / reflux; 2: With hydrogenchloride in tetrahydrofuran; water 3 h; Heating / reflux; 3: With sodium hydroxide in tetrahydrofuran; water
参考文献
GENERICS [UK] LIMITED; MERCK DEVELOPMENT CENTRE PRIVATE LIMITED
Patent: WO2008/93142 A1, 2008 ;
Location in patent: Page/Page column title page; 12; Sheet 3/3 ;