反应条件
1: in N,N-dimethyl-formamide
T=30°C; 1 h;
2: With acetic anhydride in N,N-dimethyl-formamide
T=80°C; 16 h;
参考文献
Buller, Fabian; Mannocci, Luca; Zhang, Yixin; Dumelin, Christoph E.; Scheuermann, Joerg; Neri, Dario
Bioorganic and Medicinal Chemistry Letters, 2008 , vol. 18, # 22 p. 5926 - 5931