反应条件
1: With sodium methylate in 1,4-dioxane; methanol T=5 - 15°C; Inert atmosphere; 2: With ammonia in 1,4-dioxane; methanol T=20°C; 2 h; Inert atmosphere;
参考文献
Frutos, Rogelio P.; Wei, Xudong; Patel, Nitinchandra D.; Tampone, Thomas G.; Mulder, Jason A.; Busacca, Carl A.; Senanayake, Chris H.
Journal of Organic Chemistry, 2013 , vol. 78, # 11 p. 5800 - 5803