1: 2-Chloro-1H-1,3-benzimidazole With sodium hydride in N,N-dimethyl-formamide
2: 1-(chloromethyl)-4-(trifluoromethyl)benzene in N,N-dimethyl-formamide
T=20°C; Further stages.;
参考文献
Da Settimo; Boldrini; Primofiore; La Motta; Taliani; Simorini; Novellino; Greco; Lavecchia
Journal of Medicinal Chemistry, 2001 , vol. 44, # 25 p. 4359 - 4369