反应条件
1: 1.) NH4Cl, Zn, 2.) NaHCO3 / 1.) DMF, 0 deg C, 1.5 h, 2.) Et2O, 0 deg C, 1 h
2: HCl / H2O / pH 4-5
View Scheme
参考文献
Marhevka, Virginia C.; Ebner, Nancy A.; Sehon, Russell D.; Hanna, Patrick E.
Journal of Medicinal Chemistry, 1985 , vol. 28, # 1 p. 18 - 24