1: 2-amino-thiazole; 1,1'-carbonyldiimidazole With 4-(N,N-dimethlyamino)pyridine in dichloromethane
T=20°C; 1 h;
2: N,N-dicyclopentylamine in dichloromethane
T=20°C;
参考文献
NOVO NORDISK A/S
Patent: WO2007/6760 A1, 2007 ;
Location in patent: Page/Page column 114 ;
WO 2007/006760 A1