1: 2-(5-bromo-1H-indol-3-yl)acetic acid With lithium hexamethyldisilazane in tetrahydrofuran
T=-78°C; 1 h;
2: benzyl chloroformate in tetrahydrofuran
T=-78°C; 2 h;
参考文献
CENTRE NATIONAL DE LA RECHERCHE SCIENTIFIQUE (CNRS); UNIVERSITE RENE DESCARTES (PARIS V)
Patent: EP1683521 A1, 2006 ;
Location in patent: Page/Page column 10; 14 ;
EP 1683521 A1